Methoxetamine

pharmacological · nervous · renal · Oral · Intranasal · Intramuscular · Sublingual

Methoxetamine. Ketamine analog (arylcyclohexylamine) dissociative; an NMDA-receptor antagonist with additional serotonin-transporter activity, giving a longer and…

Ketamine analog (arylcyclohexylamine) dissociative; an NMDA-receptor antagonist with additional serotonin-transporter activity, giving a longer and more potent dissociative experience than ketamine. Associated with ketamine-like bladder/renal toxicity and a higher overdose risk from its long duration.

PubChem CID 52911279. NMDA occupancy + t½ deferred to enrichment pass.