Tolterodine

pharmacological · digestive · renal · Oral

Tolterodine. Bladder-preferential M3 muscarinic antagonist — designed for higher detrusor selectivity vs salivary gland. Active 5-OH metabolite via CYP2D6. Slightly…

Bladder-preferential M3 muscarinic antagonist — designed for higher detrusor selectivity vs salivary gland. Active 5-OH metabolite via CYP2D6. Slightly cleaner anticholinergic profile than oxybutynin, but still meaningful Beers-list concerns.

Sources: PMID:9630826, PMID:9247842, PMID:11327200, PMID:10206324