Serotonin receptor pharmacology

receptor_pharmacology · nervous · digestive · cardiovascular

Serotonin receptor pharmacology. 5-HT1/2/3/4/6/7 + SERT. Receptor pharmacology pathway. 5-HT family receptors (all GPCR except 5-HT3 which is a ligand-gated cation…

Modulators

• fluoxetine — inhibitor
• sertraline — inhibitor
• paroxetine — inhibitor
• citalopram — inhibitor
• escitalopram — inhibitor
• fluvoxamine — inhibitor
• venlafaxine — inhibitor
• duloxetine — inhibitor
• vortioxetine — inhibitor
• sumatriptan — activator

Sources: PMID:26841800, PMID:10462127