GABA-B receptor signaling

receptor_pharmacology · nervous

GABA-B receptor signaling. metabotropic Gi/o. Receptor pharmacology pathway. GABA-B receptors are the metabotropic arm of GABAergic inhibition: obligate heterodimers…

Modulators

• baclofen — activator
• phenibut — activator
• ghb — activator
• gaba — substrate

Sources: PMID:15269338, PMID:12037141, PMID:22595784, PMID:20655485, PMID:8532848